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1  -  30   to   730   items

     
    Ligand - Based virtual screening procedure for the prediction and the identification of novel β-amyloid aggregation inhibitors using Kohonen maps and Counterpropagation Artificial Neural Networks
    Creator: Melagraki, G, Kollias, G, Koutentis, PA, Sarimveis, H, Afantitis, A
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2011
    Language: English
    Journal: European Journal of Medicinal Chemistry
    Institution: National Technical University of Athens
    Collection : Digital Library of National Technical University of Athens | Dspace@NTUA
    RDF

    Synthesis and evaluation of the antioxidant and anti-inflammatory activity of novel coumarin-3-aminoamides and their alpha-lipoic acid adducts
    Creator: Melagraki, G, Koufaki, M, Kontogiorgis, C, Detsi, A, Hadjipavlou-Litina, DJ, Igglessi-Markopoulou, O, Afantitis, A
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2009
    Language: English
    Journal: European Journal of Medicinal Chemistry
    Institution: National Technical University of Athens
    Collection : Digital Library of National Technical University of Athens | Dspace@NTUA
    RDF

    A novel QSAR model for predicting the inhibition of CXCR3 receptor by 4-N-aryl-[1,4] diazepane ureas
    Creator: Melagraki, G, Kollias, G, Sarimveis, H, Igglessi-Markopoulou, O, Afantitis, A
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2009
    Language: English
    Journal: European Journal of Medicinal Chemistry
    Institution: National Technical University of Athens
    Collection : Digital Library of National Technical University of Athens | Dspace@NTUA
    RDF

    Design and synthesis of novel quinolinone-3-aminoamides and their alpha-lipoic acid adducts as antioxidant and antiiflammatory agents
    Creator: Koufaki, M, Melagraki, G, Prousis, KC, Kontogiorgis, C, Detsi, A, Hadjipavlou-Litina, DJ, Igglessi-Markopoulou, O, Athanasellis, G, Afantitis, A, Bouloumbasi, D
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2007
    Language: English
    Journal: JOURNAL OF MEDICINAL CHEMISTRY
    Institution: National Technical University of Athens
    Collection : Digital Library of National Technical University of Athens | Dspace@NTUA
    RDF

    Σχεδιασμός και σύνθεση νέων υποκατεστημένων πυραζολοπυριδινών ως πιθανών αναστολέων προτεϊνικών κινασών The design and synthesis of new substituted pyrazolopyridines as potential inhibitors of protein ninases
    Creator: Giannouli, Vassiliki, Γιαννούλη, Βασιλική
    Item type: PhD thesis
    Scientific field: Medicinal chemistry
    Υear: 2013
    Language: Greek
    School/department/institute: National and Kapodistrian University of Athens ▶ School of Health Sciences ▶ Department of Pharmacy ▶ Section of Pharmaceutical Chemistry
    Institution: National Documentation Centre (EKT)
    Collection : National Archive of PhD Theses  | ΕΚΤ NA.Ph.D.
    RDF

    Επίδραση της ολευρωπαΐνης στην χρόνια καρδιακή ανεπάρκεια που προκαλεί η χορήγηση της αδριαμυκίνης: μελέτη του μηχανισμού δράσης Effect of oleuropein in adriamycin induced heart failure: study of the mechanism of action
    Creator: Ioannidis, Konstantinos, Ιωαννίδης, Κωνσταντίνος
    Item type: PhD thesis
    Scientific field: Medicinal chemistry
    Υear: 2012
    Language: Greek
    School/department/institute: National and Kapodistrian University of Athens ▶ School of Health Sciences ▶ Department of Pharmacy ▶ Section of Pharmaceutical Chemistry
    Institution: National Documentation Centre (EKT)
    Collection : National Archive of PhD Theses  | ΕΚΤ NA.Ph.D.
    RDF

    Σχεδιασμός και σύνθεση πουρινικών αναλόγων που φέρουν ομάδες νιτρικών εστέρων: φαρμακολογική μελέτη της καρδιοπροστατευτικής τους δράσης Design and synthesis of purine analogues bearing nitrate esters: pharmacological study of their cardioprotective activity
    Creator: Fotopoulou, Theano, Φωτοπούλου, Θεανώ
    Item type: PhD thesis
    Scientific field: Medicinal chemistry
    Υear: 2011
    Language: Greek
    School/department/institute: National and Kapodistrian University of Athens ▶ School of Health Sciences ▶ Department of Pharmacy ▶ Section of Pharmaceutical Chemistry
    Institution: National Documentation Centre (EKT)
    Collection : National Archive of PhD Theses  | ΕΚΤ NA.Ph.D.
    RDF

    Σύμπλοκα του τεχνητίου και του ρηνίου με πιθανό φαρμακολογικό ενδιαφέρον
    Creator: Παπαχρίστου, Μαρία, Papachristou, Maria
    Item type: PhD thesis
    Scientific field: Medicinal chemistry
    Υear: 2002
    Language: Greek
    School/department/institute: National and Kapodistrian University of Athens ▶ School of Health Sciences ▶ Department of Pharmacy ▶ Section of Pharmaceutical Chemistry
    Institution: National Documentation Centre (EKT)
    Collection : National Archive of PhD Theses  | ΕΚΤ NA.Ph.D.
    RDF

    Σπειροκαρβοκυκλικά και αρυλοϋποκατεστημένα 2,6-δικετοπιπεραζινο-1-ακετοϋδροξαμικά και σπειροκαρβοκυκλικά Ν-[(2,6-δικετοπιπεραζιν-1-υλ)ακετυλο] γλυκινοϋδροξαμικά οξέα: σχεδιασμός, σύνθεση και αξιολόγηση της αντιτυπανοσωμιακής in vitro δράσης Spirocarbocyclic and aryl-substituted 2,6-diketopiperazino-1-acetohydroxamic and spirocarbocyclic N-[(2,6-diketopiperazin-1-yl)acetyl]glycinehydroxamic acids: design, synthesis and evaluation of their in vitro antitrypanosomal activity
    Creator: Tsatsaroni, Alexandra, Τσατσαρώνη, Αλεξάνδρα
    Item type: PhD thesis
    Scientific field: Medicinal chemistry
    Υear: 2016
    Language: Greek
    School/department/institute: National and Kapodistrian University of Athens ▶ School of Health Sciences ▶ Department of Pharmacy ▶ Section of Pharmaceutical Chemistry
    Institution: National Documentation Centre (EKT)
    Collection : National Archive of PhD Theses  | ΕΚΤ NA.Ph.D.
    RDF

    Δομικές μελέτες των ογκοπρωτεϊνών c-Myc και PI3Kα και ανάπτυξη νέων συνθετικών μορίων που αναστέλουν τη δράση τους
    Creator: Ευαγγελίδης, Θωμάς, Evangelidis, Thomas
    Item type: PhD thesis
    Scientific field: Medicinal chemistry
    Υear: 2017
    Language: English
    School/department/institute: National and Kapodistrian University of Athens ▶ School of Health Sciences ▶ Department of Pharmacy ▶ Section of Pharmaceutical Chemistry
    Institution: National Documentation Centre (EKT)
    Collection : National Archive of PhD Theses  | ΕΚΤ NA.Ph.D.
    RDF

    Συγκριτική συνεισφορά φύλλων, ανθέων και άλλων φυτικών οργάνων στην απόδοση σε αιθέριο έλαιο του Orıganum vulgare spp hırtum
    Creator: Αντωνιάδου, Άννα
    Item type: Bachelor thesis
    Scientific field: Medicinal chemistry
    Language: Greek
    Institution: University of Ioannina
    Collection : Repository of UOI Olympias
    RDF

    Συγκριτική συνεισφορά φύλλων ανθέων και άλλων φυτικών οργάνων στην απόδοση σε αιθέριο έλαιο του Origanum vulgare spp hirtum.
    Creator: Αντωνιάδου, Άννα
    Item type: Bachelor thesis
    Scientific field: Medicinal chemistry
    Υear: 2017
    Institution: University of Ioannina
    Collection : Repository of UOI Olympias
    RDF

    Τα αιθέρια έλαια στη φυτοπροστασία.
    Creator: Δήμος, Αναστάσιος
    Item type: Bachelor thesis
    Scientific field: Medicinal chemistry
    Υear: 2015
    Language: Greek
    Institution: University of Ioannina
    Collection : Repository of UOI Olympias
    RDF

    Μελέτη της απόδοσης σε αιθέριο έλαιο του sideritis perfoliate σε συνθήκες καλλιέργειας.
    Creator: Τσακανίκας, Ευάγγελος
    Item type: Bachelor thesis
    Scientific field: Medicinal chemistry
    Language: Greek
    Institution: University of Ioannina
    Collection : Repository of UOI Olympias
    RDF

    Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
    Creator: Mangani S., Kebede B., Behrens B., Iacono L.D., Linciano P., Pozzi C., Reinshagen J., Borsari C., Corral M.J., Santucci M., Costi M.P., Uliassi E., Landi G., Quotadamo A., Bolognesi M.L., Di Pisa F., Venturelli A., Santarem N., Karunakaran D., Wolf M., Pöhner I., Panecka-Hofman J., Προύσης, Κυριάκος, Fenske M., Wrigley S., Clos J., Freitas-Junior L.H., Alunda J.M., Ellinger B., Keminer O., dos Santos Pascoalino B., Cordeiro-da-Silva A., Müller W., Witt G., Gul S., Kuzikov M., Wade R.C., Moraes C.B., Bertolacini C.P., Καλογεροπούλου, Θεοδώρα, Leu J., Ferrari S.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2019
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Formulation and Structural Study of a Biocompatible Water-in-Oil Microemulsion as an Appropriate Enzyme Carrier: The Model Case of Horseradish Peroxidase
    Creator: Ζουμπανιώτη, Μαρία, Ξενάκης, Αριστοτέλης, Georgiou D., Mitsou E., Kalogianni E.P., Stamatis H.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2019
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Impact of antioxidant natural compounds on the thyroid gland and implication of the Keap1/Nrf2 signaling pathway
    Creator: Paunkov A., Χονδρογιάννη, Νίκη, Chartoumpekis D.V., Ziros P.G., Kensler T.W., Sykiotis G.P.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2019
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Synergistic combination of alkylphosphocholines with peptaibols in targeting Leishmania infantum in vitro
    Creator: Fragiadaki I., Brückner H., Katogiritis A., Scoulica E., Καλογεροπούλου, Θεοδώρα
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2018
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    In vitro inflammatory/anti-inflammatory effects of nitrate esters of purines
    Creator: Fotopoulou T., Κουφάκη, Μαρία, Dutartre P., Maugé L., Connat J.-L., Delemasure S.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2014
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Design and synthesis of 21-alkynylaryl pregnenolone derivatives and evaluation of their anticancer activity
    Creator: Mavrofrydi O., Pantzou A., Szalóki G., Προύσης, Κυριάκος, Papazafiri P., Καλογεροπούλου, Θεοδώρα
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2014
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    A steroidal Na+/K+M ATpase inhibitor triggers pro-apoptotic signaling and induces apoptosis in prostate and lung tumor cells
    Creator: Al-Vahya H., Liu G., Dimas K., Alkahtani S., Kounenidakis M., Honisch S., Lang F., Προύσης, Κυριάκος, Stournaras C., Alarifi S., Καλογεροπούλου, Θεοδώρα, Alevizopoulos K., Alkahtane A.A., Al-Dahmash B.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2014
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Different extraction methodologies and their influence on the bioactivity of the wild edible mushroom Laetiporus sulphureus (Bull.) Murrill
    Creator: Proestos C., Papandreou M., Baskakis C., Petrović J., Soković M., Ćirić A., Ζουμπουλάκης, Παναγιώτης, Glamočlija J., Lamari F.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2014
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Structure-based design of inhibitors of the aspartic protease endothiapepsin by exploiting dynamic combinatorial chemistry
    Creator: Park A., Radeva N., Hirsch A.K.H., Klebe G., Potamitis C., Mondal M., Köster H., Ζερβού, Μαρία
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2014
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Elucidation of conformational states, dynamics, and mechanism of binding in human κ-opioid receptor complexes
    Creator: Παπαδόπουλος, Μάνθος Γ., Durdagi S., Yurtsever M., Avramopoulos A., Leonis G., Salmas R.E.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2014
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Vitamin E derivatives: A patent review (2010 - 2015)
    Creator: Κουφάκη, Μαρία
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2016
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Leveraging NMR and X-ray data of the free ligands to build better drugs targeting angiotensin II Type 1 G-Protein coupled receptor
    Creator: Liapakis G., Durdagi S., Ntountaniotis D., Tzakos A.G., Ergun G., Potamitis C., Gokdemir E., Μαυρομούστακος, Θωμάς, Kellici T.F., Kritsi E., Halabalaki M., Ζουμπουλάκης, Παναγιώτης, Gerothanassis I.P., Ζερβού, Μαρία, Salmas R.E.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2016
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Total phenolic content, antioxidant capacity and phytochemical profiling of grape and pomegranate wines
    Creator: Proestos C., Sinanoglou V.J., Lantzouraki D.Z., Ζουμπουλάκης, Παναγιώτης, Tsiaka T.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2015
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    Discovery of HIV Type 1 Aspartic Protease Hit Compounds through Combined Computational Approaches
    Creator: Xanthopoulos D., Παπαδόπουλος, Μάνθος Γ., Kritsi E., Leonis G., Ζουμπουλάκης, Παναγιώτης, Supuran C.T.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2016
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    2-Oxoamide inhibitors of cytosolic group IVA phospholipase A2with reduced lipophilicity
    Creator: Nikolaou A., Kokotos G., Αντωνοπούλου, Γεωργία, Magrioti V., Mouchlis V.D., Kokotou M.G., Dennis E.A., Barbayianni E.
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2016
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

    BNN27, a 17-spiroepoxy steroid derivative, interacts with and activates p75 neurotrophin receptor, rescuing cerebellar granule neurons from apoptosis
    Creator: Xanthopoulos K.P., Charalampopoulos I., Pediaditakis I., Προύσης, Κυριάκος, Potamitis C., Καλογεροπούλου, Θεοδώρα, Kourgiantaki A., Gravanis A., Ζερβού, Μαρία
    Item type: Scientific article, Publication in journal
    Scientific field: Medicinal chemistry
    Υear: 2016
    Language: English
    School/department/institute: National Hellenic Research Foundation ▶ Institute of Chemical Biology (2012 - ...)
    Institution: National Hellenic Research Foundation (NHRF)
    Collection : Helios - Repository of the National Hellenic Research Foundation (NHRF)  | repositories EKT
    RDF

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